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Mequitazine

CAS No. 29216-28-2

Mequitazine ( Mequitazine; Primalan; Mircol; Metaplexan )

产品货号. M18376 CAS No. 29216-28-2

Mequitazine is an effective, nonsedative and long-acting histamine H1 antagonist.

纯度: 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥340 有现货
10MG ¥470 有现货
25MG ¥737 有现货
50MG ¥1004 有现货
100MG ¥1264 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    Mequitazine
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Mequitazine is an effective, nonsedative and long-acting histamine H1 antagonist.
  • 产品描述
    Mequitazine is a potent histamine H1 antagonist or antihistamine. It competes with histamine for the normal H1-receptor sites on effector cells of the gastrointestinal tract, blood vessels and respiratory tract. Mequitazine provides effective, temporary relief of sneezing, watery and itchy eyes, and runny nose due to hay fever and other upper respiratory allergies.
  • 同义词
    Mequitazine; Primalan; Mircol; Metaplexan
  • 通路
    Others
  • 靶点
    Other Targets
  • 受体
    H1 receptor
  • 研究领域
    Inflammation/Immunology
  • 适应症
    ——

化学信息

  • CAS Number
    29216-28-2
  • 分子量
    322.47
  • 分子式
    C20H22N2S
  • 纯度
    98%
  • 溶解度
    DMSO : 16 mg/mL 49.62 mM;
  • SMILES
    C(C1CN2CCC1CC2)N1c2ccccc2Sc2ccccc12
  • 化学全称
    10-(1-azabicyclo[2.2.2]octan-3-ylmethyl)phenothiazine

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1. Gonnot V, et al. Expedient synthesis of mequitazine an antihistaminic drug by palladium catalyzed allylic alkylation of sodium phenothiazinate. Chem Pharm Bull (Tokyo). 2009 Nov;57(11):1300-2.
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