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MSC2504877

CAS No. 1460286-21-8

MSC2504877 ( 3-(4-(2-Hydroxypropan-2-yl)phenyl)-6-methylpyrrolo[1,2-a]pyrazin-1(2H)-one )

产品货号. M28544 CAS No. 1460286-21-8

MSC2504877 is an inhibitor of tankyrase and enhances the effects of clinical CDK4/6 inhibitors. MSC2504877 suppresses the upregulation of Cyclin D2 and Cyclin E2 caused by palbociclib and enhances the suppression of phospho-Rb.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥1239 有现货
10MG ¥1968 有现货
25MG ¥3831 有现货
50MG ¥5613 有现货
100MG ¥8003 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    MSC2504877
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    MSC2504877 is an inhibitor of tankyrase and enhances the effects of clinical CDK4/6 inhibitors. MSC2504877 suppresses the upregulation of Cyclin D2 and Cyclin E2 caused by palbociclib and enhances the suppression of phospho-Rb.
  • 产品描述
    MSC2504877 is an inhibitor of tankyrase and enhances the effects of clinical CDK4/6 inhibitors. MSC2504877 suppresses the upregulation of Cyclin D2 and Cyclin E2 caused by palbociclib and enhances the suppression of phospho-Rb.
  • 同义词
    3-(4-(2-Hydroxypropan-2-yl)phenyl)-6-methylpyrrolo[1,2-a]pyrazin-1(2H)-one
  • 通路
    Others
  • 靶点
    Other Targets
  • 受体
    PTP1B
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    1460286-21-8
  • 分子量
    282.3
  • 分子式
    C17H18N2O2
  • 纯度
    >98% (HPLC)
  • 溶解度
    ——
  • SMILES
    O=C1NC(=CN2C1=CC=C2C)C=3C=CC(=CC3)C(O)(C)C
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Steinhauer J, et al. Drosophila lysophospholipid acyltransferases are specifically required for germ cell development. Mol Biol Cell. 2009 Dec;20(24):5224-35.
产品手册
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