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MGH-CP1

CAS No. 896657-58-2

MGH-CP1 ( —— )

产品货号. M24919 CAS No. 896657-58-2

MGH-CP1 is a potent and selective inhibitor TEAD palmitoylation. It exhibits dose-dependent and potent inhibition of TEAD2/4 auto-palmitoylation in vitro with IC50 of 710 nM and 672 nM, respectively.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
2MG ¥275 有现货
5MG ¥446 有现货
10MG ¥721 有现货
25MG ¥1596 有现货
50MG ¥2811 有现货
100MG ¥4560 有现货
500MG ¥9558 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    MGH-CP1
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    MGH-CP1 is a potent and selective inhibitor TEAD palmitoylation. It exhibits dose-dependent and potent inhibition of TEAD2/4 auto-palmitoylation in vitro with IC50 of 710 nM and 672 nM, respectively.
  • 产品描述
    MGH-CP1 is a potent and selective inhibitor TEAD palmitoylation. It exhibits dose-dependent and potent inhibition of TEAD2/4 auto-palmitoylation in vitro with IC50 of 710 nM and 672 nM, respectively.
  • 同义词
    ——
  • 通路
    Others
  • 靶点
    Other Targets
  • 受体
    TEAD;TEAD2;TEAD4
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    896657-58-2
  • 分子量
    368.5
  • 分子式
    C20H24N4OS
  • 纯度
    >98% (HPLC)
  • 溶解度
    DMSO:74 mg/mL (200.81 mM);Ethanol:74 mg/mL (200.81 mM)
  • SMILES
    C1C2CC3CC1CC(C2)(C3)C4=CC=C(C=C4)NC(=O)CSC5=NC=NN5
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Li Q , Sun Y , Jarugumilli G K , et al. Lats1/2 Sustain Intestinal Stem Cells and Wnt Activation through TEAD-Dependent and Independent Transcription[J]. Cell stem cell, 2020.
产品手册
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