Boeravinone B, a novel efflux pump inhibitor, apart from inhibiting the MdeA mediated efflux, also significantly inhibit the biofilm formation of S. aureus, boeravinone B may be used in combination with mupirocin for further development.

Sempervirine nitrate , a specific molecular inhibitor of Mdm2, to MEF cells abrogated Period 2 ubiquitination leading to the accumulation of a stable pool of Period 2.

FATP1-IN-1 (compound 5k) 是一种脂肪酸转运蛋白 1(FATP1) 抑制剂。FATP1-IN-1 抑制重组人或小鼠 FATP1 acyl-CoA 合成酶活性，IC50 值分别为 0.046 μM和 0.60 μM。