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Estrone O-sulfamate
CAS No. 148672-09-7
Estrone O-sulfamate ( —— )
产品货号. M36460 CAS No. 148672-09-7
Estrone O-sulfamate (Estrone 3-O-sulfamate) 是一种有效的类固醇硫酸酯酶 (STS) 抑制剂。Estrone O-sulfamate 对胎盘微粒体 (P.M.) 制剂和 MCF-7 细胞中的 STS 具有抑制活性，IC50 值分别为 18 nM 和 0.83 nM。Estrone O-sulfamate 可用于癌症的研究。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥1577 | 有现货 |
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| 10MG | ￥2328 | 有现货 |
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| 25MG | ￥3376 | 有现货 |
|
| 50MG | ￥4566 | 有现货 |
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| 100MG | ￥5967 | 有现货 |
|
| 200MG | ￥8001 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Estrone O-sulfamate
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Estrone O-sulfamate (Estrone 3-O-sulfamate) 是一种有效的类固醇硫酸酯酶 (STS) 抑制剂。Estrone O-sulfamate 对胎盘微粒体 (P.M.) 制剂和 MCF-7 细胞中的 STS 具有抑制活性，IC50 值分别为 18 nM 和 0.83 nM。Estrone O-sulfamate 可用于癌症的研究。
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产品描述Estrone O-sulfamate (Estrone 3-O-sulfamate) is a potent steroid sulfatase (STS) inhibitor. Estrone O-sulfamate has inhibitory activity for STS in a placental microsomes (P.M.) preparation and in MCF-7 cells with IC50 values of 18 nM and 0.83 nM, respectively. Estrone O-sulfamate can be used for the research of cancer.
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体外实验Estrone O-sulfamate (Estrone 3-O-sulfamate) has inhibitory activity for STS in a placental microsomes (P.M.) preparation and in MCF-7 cells with IC50 values of 18 nM and 0.83 nM, respectively.
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体内实验——
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同义词——
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通路Others
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靶点Other Targets
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受体Others
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研究领域——
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适应症——
化学信息
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CAS Number148672-09-7
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分子量349.44
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分子式C18H23NO4S
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纯度>98% (HPLC)
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溶解度——
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SMILESC[C@@]12[C@]([C@]3([C@@](C=4C(CC3)=CC(OS(N)(=O)=O)=CC4)(CC1)[H])[H])(CCC2=O)[H]
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
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β-Casomorphin, human...
β-Casomorphin, human TFA (Human β-casomorphin 7 TFA) an opioid peptide that ACTS as an opioid receptor agonist.
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Cajanin
Cajanin has potential hypolipidemic effects,possibly via up-regulating the ABCA1 protein expression,subsequently resulting in increased macrophage cholesterol efflux and RCT, it can significantly improve basal glucose uptake in HepG2 cells, its improving effect is concentration dependent, it exhibits effects stronger than that of rosiglitazone, which has been used as an antidiabetic drug.
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Acuminatin
(+)-Acuminatin exerts hepatoprotective activities, perhaps by serving as a potent antioxidant. (+)-trans-Acuminatin, and (+)-cis-acuminatin show weak activity against platelet aggregation with IC50 values of 108.5 and 90.02 uM, respectively.
