DAAO抑制剂-1是一种有效的D-氨基酸氧化酶(DAAO)抑制剂(IC50: 0.12 μM)。

The Staphylococcus aureus transpeptidase Sortase A (SrtA) anchors virulence and colonization-associated surface proteins to the cell wall. SrtA selectively recognizes a C-terminal LPXTG motif. SrtA readily reacts with its native substrate Abz-LPETG-Dap(DNP)-NH2, cleaving it and catalyzing the formation of an amide bond between the carboxyl group of threonine and the amino group of cell-wall crossbridges.

Pomalidomide-PEG2-OH 能够合成用于靶向蛋白质降解的分子和 PROTAC（蛋白水解靶向嵌合体）技术。