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TGX-115

CAS No. 351071-62-0

TGX-115 ( —— )

产品货号. M34039 CAS No. 351071-62-0

TGX-115 is a cell-permeable and potent inhibitor of the PI 3-K isoform p110β/p110δ (IC50 values of 0.13 μM for p110β and 0.63 μM for p110δ), an enzyme that regulates platelet adhesion and inhibits phosphoinositide (PI) 3-kinase, and can be used to treat coronary artery occlusion, stroke, acute coronary artery It can be used to treat cardiovascular diseases such as coronary occlusion, stroke, acute coronary syndrome, acute myocardial infarction, restenosis, atherosclerosis and unstable angina.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥3202 有现货
10MG ¥4437 有现货
25MG ¥6250 有现货
50MG ¥7700 有现货
100MG ¥9450 有现货
200MG ¥12510 有现货
500MG 获取报价 有现货
1G 获取报价 有现货
1 mL x 10 mM in DMSO ¥2651 有现货

生物学信息

  • 产品名称
    TGX-115
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    TGX-115 is a cell-permeable and potent inhibitor of the PI 3-K isoform p110β/p110δ (IC50 values of 0.13 μM for p110β and 0.63 μM for p110δ), an enzyme that regulates platelet adhesion and inhibits phosphoinositide (PI) 3-kinase, and can be used to treat coronary artery occlusion, stroke, acute coronary artery It can be used to treat cardiovascular diseases such as coronary occlusion, stroke, acute coronary syndrome, acute myocardial infarction, restenosis, atherosclerosis and unstable angina.
  • 产品描述
    TGX-115 is a cell-permeable and potent inhibitor of the PI 3-K isoform p110β/p110δ (IC50 values of 0.13 μM for p110β and 0.63 μM for p110δ), an enzyme that regulates platelet adhesion and inhibits phosphoinositide (PI) 3-kinase, and can be used to treat coronary artery occlusion, stroke, acute coronary artery It can be used to treat cardiovascular diseases such as coronary occlusion, stroke, acute coronary syndrome, acute myocardial infarction, restenosis, atherosclerosis and unstable angina.
  • 体外实验
    ——
  • 体内实验
    ——
  • 同义词
    ——
  • 通路
    PI3K/Akt/mTOR signaling
  • 靶点
    PI3K
  • 受体
    PI3K
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    351071-62-0
  • 分子量
    336.38
  • 分子式
    C20H20N2O3
  • 纯度
    >98% (HPLC)
  • 溶解度
    ——
  • SMILES
    CC1=CC=CC=C1OC1=CC=CC2=C1NC(=CC2=O)N1CCOCC1
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

产品手册
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