Didesmethyl cariprazine

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断

Didesmethyl cariprazine 是 Cariprazine 的代谢物，作为主要的循环活性部分。Didesmethyl cariprazine 的半衰期较长，为 1-3 周。Cariprazine是一种新型抗精神病候选活性分子，能结合 D3, D2 和 5-HT1A 。

Didesmethyl cariprazine is a metabolite of Cariprazine and acts as the predominant circulating active moiety. Didesmethyl cariprazine has a long half-life of 1-3 weeks. Cariprazine is a antipsychotic agent candidate that exhibits high affinity for the D3 and D2 receptors, and moderate affinity for the 5-HT1A receptor.

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GPCR/G Protein

5-HT Receptor

5-HT Receptor | Dopamine Receptor

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839712-25-3

399.36

C19H28Cl2N4O

>98% (HPLC)

In Vitro:?DMSO 中的溶解度 : 11.36 mg/mL (28.45 mM; 超声助溶 (<80°C)

NC(=O)N[C@H]1CC[C@H](CCN2CCN(CC2)c2cccc(Cl)c2Cl)CC1

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(-20℃)

With Ice Pack

≥ 2 years