Escitalopram Oxalate 是一种选择性血清素 (5-HT) 再摄取抑制剂 (SSRI)，Ki 为 0.89 nM。

GSK778 hydrochloride hydrochloride is a potent and selective BD1 bromodomain inhibitor of the BET proteins, with IC50s of 75 nM (BRD2 BD1), 41 nM (BRD3 BD1), 41 nM (BRD4 BD1), and 143 nM (BRDT BD1), respectively. GSK778 hydrochloride hydrochloride phenocopies the effects of pan-BET inhibitors in cancer models.

CBP-IN-1 是 p300/CBP bromodomain 的有效抑制剂。