CGP 29030A is a new piperazine derivative with analgesic activity and significant inhibitory effect on potentially nociceptive dorsal horn neurons, which can be used to study painful disorders.

Vasopressin acetate is a peptide hormone with vasoconstrictive and antidiuretic activities that binds to the vascular arginine vasopressin receptor, V1, with Kd values of 1.31 and 1.44 nM in A7r5 rat aortic smooth muscle cells and neonatal rat cardiomyocytes, respectively

LDN-212320 是一种谷氨酸转运蛋白 EAAT2 激活剂。 24 小时后，浓度 < 5 μM 时，它还能将 EAAT2 水平提高 6 倍以上。