Naringenin triacetate exhibits a better binding affinity with multiple crystal structures of first bromodomain BRD4 (BRD4 BD1) when compared with the known inhibitors.

Cdk4/6 抑制剂 IV 是一种细胞渗透性三氨基嘧啶，可逆地阻断 Cdk4/cyclin D1 和 Cdk6/cyclin D1 活性，IC50 值分别为 1.5 和 5.6 μM。

β-Neo-Endorphin 是一种内源性阿片肽。β-Neo-Endorphin 是一种起源于猪的下丘脑“大”亮氨酸脑啡肽。β-Neo-Endorphin 可激活 Erk1/2, MMP-2 和 MMP-9。