G-Protein antagonist peptide ( —— )

产品货号. M30670 CAS No. 143675-79-0

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

G-Protein antagonist peptide
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

Substance P-related peptide that inhibits binding of G proteins to their receptors. Competitively and reversibly inhibits M2 muscarinic receptor activation of Gi or Go and inhibits Gs activation by β-adrenoceptors.
产品描述

Substance P-related peptide that inhibits binding of G proteins to their receptors. Competitively and reversibly inhibits M2 muscarinic receptor activation of Gi or Go and inhibits Gs activation by β-adrenoceptors.
体外实验

——
体内实验

——
同义词

——
通路

Others
靶点

Other Targets
受体

——
研究领域

——
适应症

——

CAS Number

143675-79-0
分子量

1093.27
分子式

C57H64N12O9S
纯度

>98% (HPLC)
溶解度

DMSO:2 mg/mL
SMILES

[H]N1[C@@H](CCC1=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@H](CC1=CNC2=C1C=CC=C2)C(=O)N[C@@H](CC1=CC=CC=C1)C(=O)N[C@H](CC1=CNC2=C1C=CC=C2)C(=O)N[C@H](CC1=CNC2=C1C=CC=C2)C(=O)N[C@@H](CCSC)C(N)=O
化学全称

——

1. Mukai et al (1992) G protein antagonists. A novel hydrophobic peptide competes with receptor for G protein binding. J.Biol.Chem. 267 16237 PMID:

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