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ICI 174,864
CAS No. 89352-67-0
ICI 174,864 ( —— )
产品货号. M30662 CAS No. 89352-67-0
Selective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称ICI 174,864
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Selective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.
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产品描述Selective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.
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体外实验——
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体内实验——
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同义词——
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通路Endocrinology/Hormones
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靶点Opioid Receptor
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受体——
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研究领域——
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适应症——
化学信息
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CAS Number89352-67-0
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分子量691.87
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分子式C38H53N5O7
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纯度>98% (HPLC)
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溶解度DMSO:69.19 mg/mL;water:1 mg/ml
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SMILESCC(C)C[C@H](NC(=O)[C@H](CC1=CC=CC=C1)NC(=O)C(C)(C)NC(=O)C(C)(C)NC(=O)[C@H](CC1=CC=C(O)C=C1)N(CC=C)CC=C)C(O)=O
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Cohen et al (1996) Opioid agonist activity of ICI 174864 and its carboxypeptidase degradation product, LY281217. J.Pharmacol.Exp.Ther. 238 769 PMID:
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