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FC131 TFA (606968-52-9 free base)
CAS No. ——
FC131 TFA (606968-52-9 free base) ( —— )
产品货号. M30047 CAS No. ——
FC131 TFA is a CXCR4 antagonist that inhibits the binding of [125I] -sdf-1 to CXCR4 with an IC50 value of 4.5 nM and has anti-hiv activity.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥972 | 有现货 |
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| 5MG | ￥2081 | 有现货 |
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| 10MG | ￥3492 | 有现货 |
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| 25MG | ￥5724 | 有现货 |
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| 50MG | ￥8136 | 有现货 |
|
| 100MG | ￥11376 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称FC131 TFA (606968-52-9 free base)
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述FC131 TFA is a CXCR4 antagonist that inhibits the binding of [125I] -sdf-1 to CXCR4 with an IC50 value of 4.5 nM and has anti-hiv activity.
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产品描述FC131 TFA is a CXCR4 antagonist that inhibits the binding of [125I] -sdf-1 to CXCR4 with an IC50 value of 4.5 nM and has anti-hiv activity.
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体外实验——
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体内实验——
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同义词——
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通路Autophagy
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靶点CXCR
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受体IC50: 4.5 nM ([125I]-SDF-1-CXCR4)
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研究领域——
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适应症——
化学信息
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CAS Number——
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分子量843.85
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分子式C38H48F3N11O8
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纯度>98% (HPLC)
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溶解度DMSO : 250 mg/mL (296.26 mM; Need ultrasonic)
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SMILES——
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化学全称Sequence:{2-Naph-Ala}-{Gly}-{Tyr}-{Arg}-{Arg}
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
Tamamura H, et al. Stereoselective synthesis of [L-Arg-L/D-3-(2-naphthyl)alanine]-type (E)-alkene dipeptide isosteres and its application to the synthesis and biological evaluation of pseudopeptide analogues of the CXCR4 antagonist FC131. J Med Chem. 2005 Jan 27;48(2):380-91.
产品手册
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