Remoxipride hydrochloride ( Roxiam | (S)-Remoxipride Hydrochloride | Remoxipride Hydrochloride Anhydrous )

产品货号. M27695 CAS No. 73220-03-8

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

Remoxipride hydrochloride
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

多巴胺 D2 受体拮抗剂。
产品描述

Dopamine D2 receptor antagonist.(In Vivo):In male Sprague-Dawley rats, Remoxipride hydrochloride (0.1-100 μM/kg; i.p.) blockes apomorphine-induced hyperactivity and dose-dependent blockades apomorphine-induced behaviors. In beagle dogs, Remoxipride hydrochloride (0.25-5 μM/kg; gavage) blockes apomorphine-induced vomiting.
体外实验

(S)-Remoxipride hydrochloride (1-100 μM; 20 min) shows binding efficiency with IC50s of ＞100, 1.57 and 42 μM for dopamine D1, dopamine D2 and α1-Adrenoccptor, respectively.
体内实验

(S)-Remoxipride hydrochloride (0.1-100 μM/kg; i.p. 60 min prior to apomorphine) blockades apomorphine-induced behaviors s in rats and vomiting in dogs.(S)-Remoxipride hydrochloride (0.1-10 mg/kg; i.p. 30 min prior to apomorphine) displaces [3H]spiperone from both striatal and extra-striatal areas.
同义词

Roxiam | (S)-Remoxipride Hydrochloride | Remoxipride Hydrochloride Anhydrous
通路

Others
靶点

Other Targets
受体

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研究领域

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适应症

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1.Richard W. Watkins, et al. Evaluation of cinnamamide as an avian repellent: Determination of a dose—response curve.

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