CP94253 hydrochloride ( CP 94253 hydrochloride )

产品货号. M27617 CAS No. 845861-39-4

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

CP94253 hydrochloride
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

CP94253 盐酸盐是一种有效的、选择性的、具有中枢活性的 5-HT1B 受体激动剂，Ki 为 2 nM。 5-HT1A、5-HT1D、5-HT1C 和 5-HT2 受体的 Ki 分别为 89、49、860 和 1600 nM。
产品描述

CP94253 hydrochloride is a potent, selective and centrally active agonist of 5-HT1B receptor with Ki of 2 nM. The Kis are 89, 49, 860, and 1600 nM for 5-HT1A, 5-HT1D, 5-HT1C and 5-HT2 receptors, respectively.
体外实验

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体内实验

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同义词

CP 94253 hydrochloride
通路

Others
靶点

Other Targets
受体

panx1|Topo IV|Bacterial|DNA-gyrase
研究领域

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适应症

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1.Poon IK, et al. Unexpected link between an antibiotic, pannexin channels and apoptosis. Nature. 2014 Mar 20;507(7492):329-34.

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