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BMS-191095
CAS No. 166095-21-2
BMS-191095 ( —— )
产品货号. M23744 CAS No. 166095-21-2
BMS-191095 是线粒体 ATP 敏感钾 (mitoKATP) 通道激活剂。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥2043 | 有现货 |
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| 10MG | ￥3069 | 有现货 |
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| 25MG | ￥4827 | 有现货 |
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| 50MG | ￥6622 | 有现货 |
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| 100MG | ￥8631 | 有现货 |
|
| 200MG | ￥11610 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
| 1 mL x 10 mM in DMSO | ￥1834 | 有现货 |
|
生物学信息
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产品名称BMS-191095
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述BMS-191095 是线粒体 ATP 敏感钾 (mitoKATP) 通道激活剂。
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产品描述BMS-191095 is mitochondrial ATP-sensitive potassium (mitoKATP) channel activator.
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体外实验——
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体内实验Animal Model:Male Wistar rats with the induction of ischemia induced by middle cerebral artery occlusion (MCAO)Dosage:2.5 or 25 μg Administration:Intraventricular infusion; 30 min/60 min/24 hours before the induction of ischemia, once Result:Reduced total infarct volume in rats with of pretreat dose of 25 mg and 24 h before MCA. Induced a rapid mitochondrial depolarization.
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同义词——
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通路Cell Cycle/DNA Damage
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靶点Potassium Channel
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受体Potassium Channel
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研究领域——
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适应症——
化学信息
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CAS Number166095-21-2
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分子量408.88
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分子式C22H21ClN4O2
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纯度>98% (HPLC)
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溶解度DMSO:90 mg/mL (220.11 mM)
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SMILESCC(C)([C@@H]([C@H]1N(Cc2ncc[nH]2)c(cc2)ccc2Cl)O)Oc(cc2)c1cc2C#N
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Katakam PV, et al. Diversity of mitochondria-dependent dilator mechanisms in vascular smooth muscle of cerebral arteries from normal and insulin-resistant rats. Am J Physiol Heart Circ Physiol. 2014 Aug 15;307(4):H493-503.
产品手册
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