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CYM2503
CAS No. 1308833-36-4
CYM2503 ( —— )
产品货号. M23466 CAS No. 1308833-36-4
CYM2503 是 GAL2 受体的正变构调节剂 (PAM)，可在体外增强甘丙肽诱导的 IP1 产生。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥872 | 有现货 |
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| 10MG | ￥1397 | 有现货 |
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| 25MG | ￥2716 | 有现货 |
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| 50MG | ￥4334 | 有现货 |
|
| 100MG | ￥5328 | 有现货 |
|
| 200MG | ￥7182 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称CYM2503
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述CYM2503 是 GAL2 受体的正变构调节剂 (PAM)，可在体外增强甘丙肽诱导的 IP1 产生。
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产品描述CYM2503 is a positive allosteric modulator (PAM) of the GAL2 receptor that potentiates galanin-induced IP1 production in vitro.?It has no affinity for the orthosteric galanin binding site of the receptor (as measured by its inability to displace iodinated galanin, or to induce IP1 accumulation on its own).
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体外实验——
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体内实验——
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同义词——
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通路GPCR/G Protein
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靶点Neuropeptide Y Receptor
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受体GAL2
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研究领域——
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适应症——
化学信息
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CAS Number1308833-36-4
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分子量777.96
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分子式C45H55N5O7
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纯度>98% (HPLC)
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溶解度DMSO:10 mM
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SMILESO=C(N[C@H](C(N[C@@H](CCCCNC(OC(C)(C)C)=O)C(NC1=CC=C(C(C)=C2)C(NC2=O)=C1)=O)=O)CC3CCCCC3)OCC4C5=CC=CC=C5C6=CC=CC=C46
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Lu X , Roberts R , Xia R , et al. GalR2-positive allosteric modulator exhibits anticonvulsant effects in animal models[J]. Proc Natl Acad Sci U S A, 2010, 107(34):15229-15234.
产品手册
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