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Pinacidil monohydrate
CAS No. 85371-64-8
Pinacidil monohydrate ( —— )
产品货号. M22560 CAS No. 85371-64-8
Pinacidil一水合物是一种钾通道激活剂、抗高血压化合物。Pinacidil水合物激活豚鼠膀胱和心脏的ATP调节的钾通道，Ki分别为104和251 nM。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥121 | 有现货 |
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| 5MG | ￥185 | 有现货 |
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| 10MG | ￥267 | 有现货 |
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| 25MG | ￥444 | 有现货 |
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| 50MG | ￥737 | 有现货 |
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| 100MG | ￥1053 | 有现货 |
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| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
| 1 mL x 10 mM in DMSO | ￥201 | 有现货 |
|
生物学信息
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产品名称Pinacidil monohydrate
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Pinacidil一水合物是一种钾通道激活剂、抗高血压化合物。Pinacidil水合物激活豚鼠膀胱和心脏的ATP调节的钾通道，Ki分别为104和251 nM。
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产品描述Pinacidil monohydrate is a potassium channel activator, antihypertensive drug.Pinacidil hydrate activates the ATP-modulated potassium channels of guinea pog bladder and heart with Ki of 104 and 251 nM, respectively.(In Vitro):Pinacidil monohydrate is a potassium channel activator. Pinacidil hydrate is an antihypertensive drug of the class of agents called "potassium channel openers". Pinacidil hydrate activates the ATP-modulated potassium channels of guinea pog bladder and heart with Ki values of 104 and 251 nM, respectively.
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体外实验Pinacidil monohydrate is a potassium channel activator. Pinacidil hydrate is an antihypertensive drug of the class of agents called "potassium channel openers". Pinacidil hydrate activates the ATP-modulated potassium channels of guinea pog bladder and heart with Ki values of 104 and 251 nM, respectively.
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体内实验——
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同义词——
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通路Cell Cycle/DNA Damage
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靶点Potassium Channel
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受体Potassium Channel
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研究领域——
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适应症——
化学信息
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CAS Number85371-64-8
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分子量263.34
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分子式C13H21N5O
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纯度>98% (HPLC)
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溶解度DMSO:97 mg/mL (368.35mM; Need ultrasonic); Ethanol:47 mg/mL (178.48mM; Need ultrasonic)
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SMILESO.CC(N\C(NC#N)=N\c1ccncc1)C(C)(C)C
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Gollasch M, et al. Pinacidil relaxes porcine and human coronary arteries by activating ATP-dependent potassium channels in smooth muscle cells. J Pharmacol Exp Ther. 1995 Nov;275(2):681-92.
产品手册
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