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A2764 dihydrochloride
CAS No. 861038-72-4
A2764 dihydrochloride ( —— )
产品货号. M21057 CAS No. 861038-72-4
A2764 diHClide 是一种高度选择性的 TRESK 抑制剂。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥354 | 有现货 |
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| 10MG | ￥568 | 有现货 |
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| 25MG | ￥958 | 有现货 |
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| 50MG | ￥1590 | 有现货 |
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| 100MG | ￥2277 | 有现货 |
|
| 200MG | ￥3231 | 有现货 |
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| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
| 1 mL x 10 mM in DMSO | ￥387 | 有现货 |
|
生物学信息
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产品名称A2764 dihydrochloride
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述A2764 diHClide 是一种高度选择性的 TRESK 抑制剂。
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产品描述A2764 dihydrochloride is a highly selective inhibitor of TRESK.
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体外实验A2764 (100 μM) inhibits the background K+ current by 42.8±11.5% when it applies to the oocytes expressing mTRESK.A2764 (100 μM) shows an improvedinhibitory potency for activated channel with an IC50 of activated channel in ionomycin-activated mTRESK current.The subsequent application of A2764 strongly inhibits the current (77.8±3.5%).A2764 (100 μM) inhibits the current of TRESK under resting conditions and in the activated state by 42.8±11.5% and 77.8±3.5%, respectively.
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体内实验——
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同义词——
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通路Cell Cycle/DNA Damage
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靶点Potassium Channel
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受体mTRESK channel
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研究领域——
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适应症——
化学信息
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CAS Number861038-72-4
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分子量351.7
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分子式C15H21Cl3N2O
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纯度>98% (HPLC)
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溶解度DMSO:41.67 mg/mL?(118.48 mM)
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SMILESCCN(CC)CCOc1ccc(Cl)c2cccnc12.Cl.Cl
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Chemically Modified Derivatives of the Activator Compound Cloxyquin Exert Inhibitory Effect on TRESK (K2P18.1) Background Potassium Channel.[J]. Molecular pharmacology 2019.
产品手册
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