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Dermorphin TFA
CAS No. 78331-26-7
Dermorphin TFA ( —— )
产品货号. M21054 CAS No. 78331-26-7
Dermorphin TFA 是一类新型阿片类肽。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥1321 | 有现货 |
|
| 5MG | ￥1881 | 有现货 |
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| 10MG | ￥2831 | 有现货 |
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| 25MG | ￥4576 | 有现货 |
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| 50MG | ￥6398 | 有现货 |
|
| 100MG | ￥8523 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Dermorphin TFA
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Dermorphin TFA 是一类新型阿片类肽。
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产品描述Dermorphin TFA is a new class of opioids-like peptides.
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体外实验Dermorphin, a peptide isolated from the skin of Phyllomedusa frogs and the peptide receptor (NOP) component by the endogenous agonist nociceptin/orphanin FQ (N/OFQ). In displacement binding studies at CHOhMu, Dermorphin and DeNo displac the binding of [3H]-DPN in a concentration dependent and saturable manner. Dermorphin displays an affinity of 7.17, while N/OFQ fails to displace [3H]-DPN at the Delta receptor. Dermorphin and DeNo stimulate the binding of GTPγ[35S] in a concentration dependent and saturable manner at the Mu receptor.
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体内实验——
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同义词——
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通路Others
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靶点Other Targets
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受体Others
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研究领域——
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适应症——
化学信息
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CAS Number78331-26-7
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分子量916.89
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分子式C42H51F3N8O12
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纯度>98% (HPLC)
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溶解度——
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SMILESC[C@@H](NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)NCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CO)C(N)=O.O=C(O)C(F)(F)F
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Castiglione R D Faoro F Perseo G et al. SYNTHESIS OF DERMORPHINS A NEW CLASS OF OPIATE-LIKE PEPTIDES[J]. Chemical Biology & Drug Design 1981 17(2):263-272.
产品手册
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