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Adrenorphin(3TFA)
CAS No. 88377-68-8
Adrenorphin(3TFA) ( Metorphamide )
产品货号. M21026 CAS No. 88377-68-8
Adrenorphin(3TFA) 是 μ-阿片受体 (Ki :12 nM) 的激动剂。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥1843 | 有现货 |
|
| 10MG | ￥2746 | 有现货 |
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| 25MG | ￥4594 | 有现货 |
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| 50MG | ￥6910 | 有现货 |
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| 100MG | ￥10080 | 有现货 |
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| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
| 1 mL x 10 mM in DMSO | ￥2964 | 有现货 |
|
生物学信息
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产品名称Adrenorphin(3TFA)
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Adrenorphin(3TFA) 是 μ-阿片受体 (Ki :12 nM) 的激动剂。
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产品描述Adrenorphin(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
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体外实验Adrenorphin (Metorphamide) is a opioid octapeptide from bovine brain, acts as a potent agonist of μ-opioid receptor, with Ki of 12 nM. The binding ratios of Ki for μ-opioid receptor/Ki for δ-opioid receptor of 0.04 and of Ki for μ-opioid receptor/Ki for κ-opioid receptor of 0.46. Adrenorphin potently inhibits catecholamine secretion evoked by 10 μM nicotine in cultured human pheochromocytoma 6 cells, with an IC50 of 1.1 μM.
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体内实验——
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同义词Metorphamide
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通路Endocrinology/Hormones
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靶点Opioid Receptor
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受体μ-opioid receptor
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研究领域——
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适应症——
化学信息
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CAS Number88377-68-8
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分子量984.18
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分子式C44H69N15O9S
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纯度>98% (HPLC)
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溶解度DMSO:50 mg/mL (50.80 mM)
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SMILESCSCCC(NC(=O)C(Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)C(N)Cc1ccc(O)cc1)C(=O)NC(CCCNC(=N)N)C(=O)NC(CCCNC(=N)N)C(=O)NC(C(N)=O)C(C)C
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Miyata A Mizuno K Minamino N et al. Regional distribution of adrenorphin in rat brain: Comparative study with PH-8P[J]. Biochemical and Biophysical Research Communications 1984 120(3):1030-1036.
产品手册
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