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Bepridil hydrochloride
CAS No. 68099-86-5
Bepridil hydrochloride ( CERM 1978 )
产品货号. M20140 CAS No. 68099-86-5
Bepridil 是一种钙通道阻滞剂，还抑制 Na+/Ca2+ 交换 (NCX)、钠通道和心脏肌膜 KATP 通道。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥238 | 有现货 |
|
| 5MG | ￥396 | 有现货 |
|
| 10MG | ￥554 | 有现货 |
|
| 25MG | ￥918 | 有现货 |
|
| 50MG | ￥1376 | 有现货 |
|
| 100MG | ￥1998 | 有现货 |
|
| 200MG | ￥2997 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
| 1 mL x 10 mM in DMSO | ￥433 | 有现货 |
|
生物学信息
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产品名称Bepridil hydrochloride
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Bepridil 是一种钙通道阻滞剂，还抑制 Na+/Ca2+ 交换 (NCX)、钠通道和心脏肌膜 KATP 通道。
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产品描述Bepridil is a calcium channel blocker and also inhibits Na+/Ca2+ exchange (NCX) sodium channels and cardiac sarcolemmal KATP channels.(In Vitro):Bepridil hydrochloride is a calcium channel blocker, with antianginal activity.(In Vivo):Bepridil hydrochloride (21 mg/kg) reduces heart rate and mean arterial pressure, decreases the mean coronary vascular resistance and increases stroke volume in rats.
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体外实验Bepridil hydrochloride is a calcium channel blocker, with antianginal activity.
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体内实验Bepridil hydrochloride (21 mg/kg) reduces heart rate and mean arterial pressure, decreases the mean coronary vascular resistance and increases stroke volume in rats.
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同义词CERM 1978
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通路GPCR/G Protein
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靶点Calcium Channel
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受体Calcium Channel
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研究领域Cardiovascular Disease
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适应症Angina pectoris; Tachycardia
化学信息
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CAS Number68099-86-5
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分子量403
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分子式C24H35ClN2O
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纯度>98% (HPLC)
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溶解度DMSO: 130 mg/mL (322.58 mM)
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SMILESCl.CC(C)COCC(CN(Cc1ccccc1)c1ccccc1)N1CCCC1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Flaim SF et al. Effects of bepridil hydrochloride on cardiocirculatory dynamics coronary vascular resistance and cardiac output distribution in normal conscious rats. J Cardiovasc Pharmacol. 1988 Mar;11(3):363-72.
产品手册
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