[Leu144,Arg147]-PLP (139-151) is a mutant peptide fragment of myelin proteolipid protein (PLP), with the tryptophan and histidine at positions 144 and 147 respectively replaced by leucine and arginine. [Leu144,Arg147]-PLP (139-151) also serves as a T cell receptor (TCR) antagonist for encephalitogenic Th1 clones, blocking their activation in vitro. Furthermore, [Leu144,Arg147]-PLP (139-151) can inhibit the development of experimental autoimmune encephalomyelitis (EAE).

Baohuoside VII 是从 Herba Epimedii 中分离出的一种黄酮类化合物，具有抗骨质疏松的活性。

SAR131675 是一种有效且特异性的 VEGFR-3 抑制剂。它分别抑制 HEK 细胞中的 VEGFR-3 酪氨酸激酶活性 (IC50: 20 nmol/L) 和 VEGFR-3 自磷酸化 (IC50: 45 nmol/L)。