CFMTI ( CFMTI )

产品货号. M17627 CAS No. 864864-17-5

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

CFMTI
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

CFMTI 是一种有效的选择性代谢型谷氨酸受体 (mGluR) 1 变构拮抗剂 (IC50: 2.6 nM)。
产品描述

CFMTI is a potent and selective metabotropic glutamate receptor (mGluR) 1 allosteric antagonist (IC50: 2.6 nM). The selectivity of CFMTI to mGluR1 is higher 2000-fold than mGluR5.
体外实验

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体内实验

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同义词

CFMTI
通路

Membrane Transporter/Ion Channel
靶点

Beta Amyloid
受体

mGluR
研究领域

Cancer
适应症

——

CAS Number

864864-17-5
分子量

349.37
分子式

C19H16FN5O
纯度

>98% (HPLC)
溶解度

DMSO : 6.2 mg/mL. 17.75 mM;
SMILES

c1(c(nccc1)F)n1nnc(c1C)c1ccc2c(c1)CN(C2=O)C1CC1
化学全称

2-Cyclopropyl-5-[1-(2-fluoro-3-pyridinyl)-5-methyl-1H-1,2,3-triazol-4-yl]-2,3-dihydro-1H-isoindol-1-one

1.Satow A et al. 2009 Jul;330(1):179-90.

计算器

产品手册

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