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LGD-3303
CAS No. 917891-35-1
LGD-3303 ( LGD3303 )
产品货号. M16590 CAS No. 917891-35-1
LGD-3303 是一种口服、脑渗透性非甾体选择性雄激素受体调节剂 (SARM)，与相关核受体几乎没有或没有交叉反应。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥529 | 有现货 |
|
| 10MG | ￥794 | 有现货 |
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| 50MG | ￥2558 | 有现货 |
|
| 100MG | 获取报价 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称LGD-3303
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述LGD-3303 是一种口服、脑渗透性非甾体选择性雄激素受体调节剂 (SARM)，与相关核受体几乎没有或没有交叉反应。
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产品描述LGD-3303 is an orally available, brain-penetrant nonsteroidal selective androgen receptor modulator (SARM) that that shows little or no cross-reactivity with related nuclear receptors; has potent activity on levator ani muscle but is a partial agonist on the preputial gland and ventral prostate in a castrated rat model of androgen deficiency; enhances male-directed sexual preference, proceptive behavior, and lordosis behavior in sexually experienced, but not sexually naive, female rats.
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体外实验——
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体内实验——
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同义词LGD3303
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通路Endocrinology/Hormones
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靶点Androgen Receptor (AR)
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受体AndrogenReceptor
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研究领域——
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适应症——
化学信息
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CAS Number917891-35-1
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分子量342.743
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分子式C16H14ClF3N2O
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纯度>98% (HPLC)
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溶解度DMSO: Soluble （ < 1 mg/ml refers to the product slightly soluble or insoluble )
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SMILESO=C1NC2=C(C3=C(N(CC(F)(F)F)C(CC)=C3C)C=C2)C(Cl)=C1
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化学全称9-Chloro-2-ethyl-1-methyl-3-(2,2,2-trifluoroethyl)-3H-pyrrolo(3,2-F)quinolin-7(6H)-one
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Vajda EG, et al. J Pharmacol Exp Ther. 2009 Feb;328(2):663-70.
2. Vajda EG, et al. J Bone Miner Res. 2009 Feb;24(2):231-40.
3. Kudwa AE, et al. Endocrinology. 2010 Jun;151(6):2659-68.
产品手册
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