021-51111890
购物车（）
sales@molnova.cn
Setiptiline maleate
CAS No. 85650-57-3
Setiptiline maleate ( MO-8282 )
产品货号. M16210 CAS No. 85650-57-3
一种四环抗抑郁药 (TeCA)，充当去甲肾上腺素再摄取抑制剂、α2-肾上腺素受体拮抗剂和血清素受体拮抗剂。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥109 | 有现货 |
|
| 5MG | ￥161 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
| 1 mL x 10 mM in DMSO | ￥566 | 有现货 |
|
生物学信息
-
产品名称Setiptiline maleate
-
注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
-
产品简述一种四环抗抑郁药 (TeCA)，充当去甲肾上腺素再摄取抑制剂、α2-肾上腺素受体拮抗剂和血清素受体拮抗剂。
-
产品描述A tetracyclic antidepressant (TeCA) that acts as a norepinephrine reuptake inhibitor, α2-adrenergic receptor antagonist, and serotonin receptor antagonist, as well as an H1 receptor inverse agonist/antihistamine.Depression Approved.
-
体外实验——
-
体内实验——
-
同义词MO-8282
-
通路GPCR/G Protein
-
靶点5-HT Receptor
-
受体5-HT Receptor
-
研究领域Neurological Disease
-
适应症Depression
化学信息
-
CAS Number85650-57-3
-
分子量377.433
-
分子式C23H23NO4
-
纯度>98% (HPLC)
-
溶解度10 mM in DMSO
-
SMILESCN1CCC2=C(C1)C3=CC=CC=C3CC4=CC=CC=C24.C(=CC(=O)O)C(=O)O
-
化学全称1H-Dibenzo[3,4:6,7]cyclohepta[1,2-c]pyridine, 2,3,4,9-tetrahydro-2-methyl-, (2Z)-2-butenedioate (1:1)
运输与储存
-
储存条件(-20℃)
-
运输条件With Ice Pack
-
稳定性≥ 2 years
参考文献
1. Niho T, et al. Nihon Yakurigaku Zasshi. 1986 Oct;88(4):309-20.
2. Mizota M, et al. Nihon Yakurigaku Zasshi. 1986 Dec;88(6):457-66.
3. Przegaliński E, et al. Pol J Pharmacol Pharm. 1986 Jul-Aug;38(4):377-84.
产品手册
关联产品
-
Tropanserin
Tropanserin 是一种 5-羟色胺能活性化合物，也是 5-HT3 受体拮抗剂。Tropanserin 可调节外源性血清素挑战的心肺反射效应。
-
BF-1
BF-1 is a novel selective 5-HT2 receptor antagonist that acts by blocking neurogenic dural plasma protein extravasation induced by mCPP or BW723C86.BF-1 is used in the study of migraine.
-
Ticalopride
Ticalopride is a 5-HT3 receptor agonist used in the treatment of digestive disorders, orofacial disorders, otorhinolaryngologic disorders, and may be used in the study of bulimia nervosa, gastroesophageal reflux, and irritable bowel syndrome.
