Tetracaine hydrochloride
CAS No. 136-47-0
Tetracaine hydrochloride ( —— )
产品货号. M11504 CAS No. 136-47-0
盐酸丁卡因 (Pontocaine) 是丁卡因的盐酸盐形式,是一种有效的局部麻醉剂和通道功能变构抑制剂。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 500MG | ¥148 | 有现货 |
|
| 1G | ¥224 | 有现货 |
|
生物学信息
-
产品名称Tetracaine hydrochloride
-
注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
-
产品简述盐酸丁卡因 (Pontocaine) 是丁卡因的盐酸盐形式,是一种有效的局部麻醉剂和通道功能变构抑制剂。
-
产品描述Tetracaine hydrochloride (Pontocaine) is a hydrochloride salt form of tetracaine which is a potent local anaesthetic and a channel function allosteric inhibitor. Tetracaine hydrochloride (Pontocaine) is used to block temporarily the pain "message" that is sent along the nerves that connect the eyes to the brain. Tetracaine hydrochloride (Pontocaine) is mainly used topically in ophthalmology and as an antipruritic, and it has been used in spinal anesthesia. (In Vitro):Tetracaine hydrochloride (Amethocaine hydrochloride) is used to alter the function of calcium release channels (ryanodine receptors) that control the release of calcium from intracellular stores. Tetracaine hydrochloride is an allosteric blocker of channel function. At low concentrations, tetracaine causes an initial inhibition of spontaneous calcium release events, while at high concentrations, tetracaine blocks release completely.
-
体外实验Tetracaine hydrochloride (Amethocaine hydrochloride) is used to alter the function of calcium release channels (ryanodine receptors) that control the release of calcium from intracellular stores. Tetracaine hydrochloride is an allosteric blocker of channel function. At low concentrations, tetracaine causes an initial inhibition of spontaneous calcium release events, while at high concentrations, tetracaine blocks release completely.
-
体内实验——
-
同义词——
-
通路Membrane Transporter/Ion Channel
-
靶点Sodium Channel
-
受体Sodium Channel
-
研究领域Neurological Disease
-
适应症——
化学信息
-
CAS Number136-47-0
-
分子量300.83
-
分子式C15H24N2O2·HCl
-
纯度>98% (HPLC)
-
溶解度Ethanol: 30 mg/mL (99.72 mM); Water: 60 mg/mL (199.45 mM); DMSO: 60 mg/mL (199.45 mM)
-
SMILESCl.CCCCNC1=CC=C(C=C1)C(=O)OCCN(C)C
-
化学全称——
运输与储存
-
储存条件(-20℃)
-
运输条件With Ice Pack
-
稳定性≥ 2 years
参考文献
1.Leng T, et al. Mol Pain. 2013 Jun 10;9:27
产品手册
关联产品
-
KR-32568
KR-32568 是一种钠/氢交换器 1 (NHE-1) 抑制剂,IC50 为 230 nM。KR-32568 具有心脏保护作用。
-
Oxcarbazepine
奥卡西平在结构上是卡马西平的衍生物,在苄基甲酰胺基团上添加了一个额外的氧原子。
-
Anemoside B4
Anemomoside B4 抑制 IL-10 的分泌。
021-51111890
购物车()
sales@molnova.cn

