Litorin

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断

Litorin，一种两栖类蛙皮素衍生物，是一种蛙皮素受体 (bombesin receptor) 激动剂。Litorin 刺激平滑肌收缩，刺激胃泌素、胃酸和胰腺分泌，抑制体内实验中的营养物质。

Litorin, an amphibian bombesin peptide derivative, is an bombesin receptor agonist. Litorin stimulates the contraction of smooth muscle, stimulates gastrin, gastric acid, and pancreatic secretion, and suppresses the nutriment in vivo.

Litorin stimulates the contraction of smooth muscle, stimulates gastrin, gastric acid, and pancreatic secretion, and suppresses the nutriment in in vivo experiments.

99mTc-Litorin is developed for non-invasive imaging of tumors with overexpressed gastrin-releasing peptide receptors (GRP-R).[D-Phe1,Leu8,9]Litorin inhibits binding of 125I-[Tyr4] BN to murine Swiss 3T3 cells with a Ki of 5.1 nM.Litorin stimulates 3H-Thymidine incorporation in murine Swiss 3T3 cells with an EC50 of 2.3 nM.

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Others

Other Targets

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55749-97-8

1085.24

C51H68N14O11S

>98% (HPLC)

DMSO : 100 mg/mL (92.15 mM; ultraphonic; ) H2O : 2 mg/mL (1.84 mM; ultraphonic (<60 ℃)； (HCL ，pH=3) )

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(-20℃)

With Ice Pack

≥ 2 years