
Linrodostat
CAS No. 1923833-60-6
Linrodostat ( BMS-986205 | ONO-7701 )
产品货号. M18180 CAS No. 1923833-60-6
BMS-986205 是一种选择性吲哚胺 2, 3-双加氧酶 1 (IDO1) 抑制剂。
纯度: >98% (HPLC)






规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥421 | 有现货 |
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10MG | ¥640 | 有现货 |
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25MG | ¥1312 | 有现货 |
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50MG | ¥2203 | 有现货 |
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100MG | ¥3540 | 有现货 |
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200MG | ¥5225 | 有现货 |
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500MG | 获取报价 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称Linrodostat
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述BMS-986205 是一种选择性吲哚胺 2, 3-双加氧酶 1 (IDO1) 抑制剂。
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产品描述BMS-986205 is a selective indoleamine 2, 3-dioxygenase 1 (IDO1) inhibitor.(In Vitro):Linrodostat (0.01-100 μM; 72 hours; SKOV-3 and Jurkat clone E6-1 cells) treatment reduces the number of viable cells compared with the non-treated control. Linrodostat also induces cell death at much lower concentrations and its IC50 is 6.3 μM.
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体外实验Linrodostat (0.01-100 μM; 72 hours; SKOV-3 and Jurkat clone E6-1 cells) treatment reduces the number of viable cells compared with the non-treated control. Linrodostat also induces cell death at much lower concentrations and its IC50 is 6.3 μM. Cell Viability Assay Cell Line:SKOV-3 and Jurkat clone E6-1 cells Concentration:0.01-100 μM Incubation Time:72 hours Result:Reduced the number of viable cells compared with the non-treated control and induced cell death at much lower concentrations.
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体内实验——
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同义词BMS-986205 | ONO-7701
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通路Others
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靶点Other Targets
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受体IDO1
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研究领域Cancer
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适应症——
化学信息
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CAS Number1923833-60-6
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分子量410.91
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分子式C24H24ClFN2O
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纯度>98% (HPLC)
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溶解度DMSO : 50 mg/mL 121.68 mM; H2O : < 0.1 mg/mL
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SMILESClc1ccc(cc1)NC(=O)[C@H](C)[C@@H]2CC[C@@H](CC2)c3ccnc4ccc(F)cc34
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Lillian L. Siu, et al. Cancer Res. 2017; 77 (13 Suppl): Abstract nr CT116.
产品手册




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