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Latrepirdine

CAS No. 97657-92-6

Latrepirdine ( Latrepirdine dimebolin Dimebon )

产品货号. M17697 CAS No. 97657-92-6

Latrepirdine is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors, GluR, and 5-HT receptors, used as an antihistamine drug.

纯度: 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥348 有现货
10MG ¥697 有现货
25MG ¥1215 有现货
50MG ¥2066 有现货
100MG ¥3443 有现货
200MG ¥4755 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    Latrepirdine
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Latrepirdine is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors, GluR, and 5-HT receptors, used as an antihistamine drug.
  • 产品描述
    Latrepirdine, also known as dimebolin (sold as Dimebon), is an antihistamine drug which has been used clinically in Russia since 1983. Research is continuing in both Russia and western nations into potential applications as a neuroprotective drug to combat Alzheimer's disease and, possibly, as a nootropic as well. However, a Phase III clinical trial for Alzheimer's disease treatment failed to show any benefit.
  • 同义词
    Latrepirdine dimebolin Dimebon
  • 通路
    Others
  • 靶点
    Other Targets
  • 受体
    GluR , Histamine receptor , 5-HT
  • 研究领域
    Inflammation/Immunology
  • 适应症
    ——

化学信息

  • CAS Number
    97657-92-6
  • 分子量
    392.37
  • 分子式
    C21H25N3·2HCl
  • 纯度
    98%
  • 溶解度
    DMSO : 6.4 mg/mL. 16.31 mM;
  • SMILES
    CC1=CC2=C(C=C1)N(C3=C2CN(CC3)C)CCC4=CN=C(C=C4)C.Cl.Cl
  • 化学全称
    2,8-dimethyl-5-(2-(6-methylpyridin-3-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole hydrochloride

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1. Zhang S, et al. J Alzheimers Dis, 2010, 21(2), 389-402.
产品手册
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