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Laniquidar
CAS No. 197509-46-9
Laniquidar ( R-101933;R101933 )
产品货号. M13087 CAS No. 197509-46-9
An orally active, third-generation P-glycoprotein inhibitor that inhibits the drug efflux pump P-glycoprotein.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥9801 | 有现货 |
|
| 50MG | ￥16038 | 有现货 |
|
| 100MG | ￥20250 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Laniquidar
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述An orally active, third-generation P-glycoprotein inhibitor that inhibits the drug efflux pump P-glycoprotein.
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产品描述An orally active, third-generation P-glycoprotein inhibitor that inhibits the drug efflux pump P-glycoprotein, resulting in higher concentrations of antineoplastic agents in tumor cells that are multi-drug resistant due to the overexpression of P-glycoprotein.Breast Cancer Phase 2
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同义词R-101933;R101933
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通路Membrane Transporter/Ion Channel
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靶点P-glycoprotein
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受体P-glycoprotein
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研究领域Cancer
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适应症Breast Cancer
化学信息
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CAS Number197509-46-9
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分子量584.70
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分子式C37H36N4O3
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纯度>98% (HPLC)
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溶解度——
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SMILESO=C(C1=CN=C2N1CCC3=CC=CC=C3/C2=C4CCN(CCC5=CC=C(OCC6=NC7=CC=CC=C7C=C6)C=C5)CC\4)OC
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化学全称methyl 11-(1-(4-(quinolin-2-ylmethoxy)phenethyl)piperidin-4-ylidene)-6,11-dihydro-5H-benzo[d]imidazo[1,2-a]azepine-3-carboxylate
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. van Zuylen L, et al. Clin Cancer Res. 2000 Apr;6(4):1365-71.
2. van Zuylen L, et al. Eur J Cancer. 2002 May;38(8):1090-9.
3. Luurtsema G, et al. Nucl Med Biol. 2009 Aug;36(6):643-9.
2. van Zuylen L, et al. Eur J Cancer. 2002 May;38(8):1090-9.
3. Luurtsema G, et al. Nucl Med Biol. 2009 Aug;36(6):643-9.
产品手册
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