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LY2183240
CAS No. 874902-19-9
LY2183240 ( —— )
产品货号. M24889 CAS No. 874902-19-9
LY2183240 inhibits fatty acid amide hydrolase (FAAH) activity (IC50 = 12.4 nM). LY2183240 is a novel and highly effective blocker of anandamide uptake (IC50 = 270 pM).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥316 | 有现货 |
|
| 10MG | ￥518 | 有现货 |
|
| 25MG | ￥1077 | 有现货 |
|
| 50MG | ￥2049 | 有现货 |
|
| 100MG | ￥3208 | 有现货 |
|
| 500MG | ￥7525 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称LY2183240
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述LY2183240 inhibits fatty acid amide hydrolase (FAAH) activity (IC50 = 12.4 nM). LY2183240 is a novel and highly effective blocker of anandamide uptake (IC50 = 270 pM).
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产品描述LY2183240 inhibits fatty acid amide hydrolase (FAAH) activity (IC50 = 12.4 nM). LY2183240 is a novel and highly effective blocker of anandamide uptake (IC50 = 270 pM).
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同义词——
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通路Autophagy
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靶点Autophagy
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受体Autophagy;FAAH
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研究领域——
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适应症——
化学信息
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CAS Number874902-19-9
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分子量307.4
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分子式C17H17N5O
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纯度>98% (HPLC)
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溶解度DMSO:50 mg/mL (162.68 mM; Need ultrasonic)
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SMILESO=C(N(C)C)N1N=NN=C1CC(C=C2)=CC=C2C3=CC=CC=C3
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Dickason-Chesterfield AK, et al. Pharmacological characterization of endocannabinoid transport and fatty acid amide hydrolase inhibitors. Cell Mol Neurobiol. 2006 Jul-Aug;26(4-6):407-23.
产品手册
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