LM10
CAS No. 1316695-35-8
LM10 ( LM10; LM 10; LM-10 )
产品货号. M17944 CAS No. 1316695-35-8
Selective tryptophan 2, 3-dioxygenase (TDO) inhibitor (IC50 values are 0.62 and 2 μM for human and mouse TDO, respectively).
纯度: 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥243 | 有现货 |
|
10MG | ¥381 | 有现货 |
|
25MG | ¥786 | 有现货 |
|
50MG | ¥1401 | 有现货 |
|
100MG | ¥2714 | 有现货 |
|
200MG | ¥4269 | 有现货 |
|
500MG | ¥6820 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称LM10
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Selective tryptophan 2, 3-dioxygenase (TDO) inhibitor (IC50 values are 0.62 and 2 μM for human and mouse TDO, respectively).
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产品描述LM10 is a selective tryptophan 2,3-dioxygenase (TDO) inhibitor (IC50 values are 0.62 and 2 μM for human and mouse TDO, respectively). LM10 exhibits selectivity for TDO over IDO, MAO-A, MAO-B, and a panel of receptors and transporters. LM10 reduces growth of TDO-expressing P815 mastocytoma tumors in mice.
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同义词LM10; LM 10; LM-10
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通路Others
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靶点Other Targets
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受体TDO
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研究领域Others-Field
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适应症——
化学信息
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CAS Number1316695-35-8
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分子量229.22
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分子式C11H8FN5
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纯度98%
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溶解度——
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SMILESFc2cc3ncc(/C=C/c1nnnn1)c3cc2
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化学全称6-fluoro-3-[(E)-2-(1H-1,2,3,4-tetrazol-5-yl)ethenyl]-1H-indole
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Pilotte L,etal.Reversal of tumoral immune resistance by inhibition of tryptophan 2,3-dioxygenase.Proc Natl Acad Sci U S A. 2012 Feb 14;109(7):2497-502.
产品手册
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