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KB-R7943

CAS No. 182004-65-5

KB-R7943 ( KB-R7943 mesylate )

产品货号. M20553 CAS No. 182004-65-5

KB-R7943 mesylate is a widely used inhibitor of the reverse Na+/Ca2+ exchanger (NCXrev) with IC50 of 5.7±2.1 μM.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥405 有现货
10MG ¥518 有现货
25MG ¥1061 有现货
50MG ¥1912 有现货
100MG ¥2876 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    KB-R7943
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    KB-R7943 mesylate is a widely used inhibitor of the reverse Na+/Ca2+ exchanger (NCXrev) with IC50 of 5.7±2.1 μM.
  • 产品描述
    KB-R7943 mesylate is a widely used inhibitor of the reverse Na+/Ca2+ exchanger (NCXrev) with IC50 of 5.7±2.1 μM.
  • 同义词
    KB-R7943 mesylate
  • 通路
    Others
  • 靶点
    Other Targets
  • 受体
    Na+/Ca2+ Exchanger
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    182004-65-5
  • 分子量
    427.5
  • 分子式
    C17H21N3O6S2
  • 纯度
    >98% (HPLC)
  • 溶解度
    DMSO:27 mg/mL (63.16 mM)
  • SMILES
    CS(O)(=O)=O.NC(=N)SCCc1ccc(OCc2ccc(cc2)[N+]([O-])=O)cc1
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Brustovetsky T Brittain M K Sheets P L et al. KB-R7943 an inhibitor of the reverse Na+ /Ca2+ exchanger blocks N-methyl-D-aspartate receptor and inhibits mitochondrial complex I.[J]. British Journal of Pharmacology 2015 162(1):255-270.
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