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JNJ-63533054
CAS No. 1802326-66-4
JNJ-63533054 ( JNJ 63533054; JNJ63533054; JNJ-63533054 )
产品货号. M17383 CAS No. 1802326-66-4
JNJ-63533054 is a potent and selective agonist of hGPR139 with an EC50 = 16 nM.
纯度: 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥486 | 有现货 |
|
| 10MG | ￥737 | 有现货 |
|
| 25MG | ￥1580 | 有现货 |
|
| 50MG | ￥2803 | 有现货 |
|
| 100MG | ￥4147 | 有现货 |
|
| 500MG | ￥8748 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称JNJ-63533054
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述JNJ-63533054 is a potent and selective agonist of hGPR139 with an EC50 = 16 nM.
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产品描述JNJ 63533054 is a potent and selective GPR139 agonist (EC50 = 16 nM) that is brain and cell penetrant. JNJ 63533054 is selective for GPR139 over a panel of GPCRs, ion channels and transporters, including GPR142 and is orally bioavailable.
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同义词JNJ 63533054; JNJ63533054; JNJ-63533054
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通路Angiogenesis
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靶点Adrenergic Receptor
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受体hGPR139
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研究领域Neurological Disease
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适应症——
化学信息
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CAS Number1802326-66-4
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分子量316.78
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分子式C17H17ClN2O2
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纯度98%
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溶解度DMSO : ≥ 50 mg/mL 157.84 mM; H2O : < 0.1 mg/mL
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SMILESC[C@@H](c1ccccc1)NC(=O)CNC(=O)c1cc(ccc1)Cl
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化学全称3-Chloro-N-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]benzamide
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Dvorak CA, et al. ACS Med Chem Lett. 2015 Jul 20;6(9):1015-8.
产品手册
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