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JNJ-63533054

CAS No. 1802326-66-4

JNJ-63533054 ( JNJ 63533054; JNJ63533054; JNJ-63533054 )

产品货号. M17383 CAS No. 1802326-66-4

JNJ-63533054 is a potent and selective agonist of hGPR139 with an EC50 = 16 nM.

纯度: 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥486 有现货
10MG ¥737 有现货
25MG ¥1580 有现货
50MG ¥2803 有现货
100MG ¥4147 有现货
500MG ¥8748 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    JNJ-63533054
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    JNJ-63533054 is a potent and selective agonist of hGPR139 with an EC50 = 16 nM.
  • 产品描述
    JNJ 63533054 is a potent and selective GPR139 agonist (EC50 = 16 nM) that is brain and cell penetrant. JNJ 63533054 is selective for GPR139 over a panel of GPCRs, ion channels and transporters, including GPR142 and is orally bioavailable.
  • 同义词
    JNJ 63533054; JNJ63533054; JNJ-63533054
  • 通路
    Angiogenesis
  • 靶点
    Adrenergic Receptor
  • 受体
    hGPR139
  • 研究领域
    Neurological Disease
  • 适应症
    ——

化学信息

  • CAS Number
    1802326-66-4
  • 分子量
    316.78
  • 分子式
    C17H17ClN2O2
  • 纯度
    98%
  • 溶解度
    DMSO : ≥ 50 mg/mL 157.84 mM; H2O : < 0.1 mg/mL
  • SMILES
    C[C@@H](c1ccccc1)NC(=O)CNC(=O)c1cc(ccc1)Cl
  • 化学全称
    3-Chloro-N-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]benzamide

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1. Dvorak CA, et al. ACS Med Chem Lett. 2015 Jul 20;6(9):1015-8.
产品手册
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