JNJ-1661010
CAS No. 681136-29-8
JNJ-1661010 ( JNJ-1661010; JNJ 1661010; JNJ1661010 )
产品货号. M18990 CAS No. 681136-29-8
JNJ-1661010 is an effective and specific FAAH inhibitor (IC50: 10/ 12 nM for rat/human), shows >100-fold selectivity for FAAH-1 than FAAH-2.
纯度: 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥316 | 有现货 |
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10MG | ¥543 | 有现货 |
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25MG | ¥1158 | 有现货 |
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50MG | ¥1847 | 有现货 |
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100MG | ¥2981 | 有现货 |
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200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称JNJ-1661010
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述JNJ-1661010 is an effective and specific FAAH inhibitor (IC50: 10/ 12 nM for rat/human), shows >100-fold selectivity for FAAH-1 than FAAH-2.
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产品描述JNJ-1661010 is a selective, reversible inhibitor of fatty acid amide hydrolase (FAAH) (IC50 = 12 nM). JNJ-1661010 is a brain penetrant and active in vivo.
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同义词JNJ-1661010; JNJ 1661010; JNJ1661010
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通路Others
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靶点Other Targets
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受体FAAH (human); FAAH (rat)
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研究领域Others-Field
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适应症——
化学信息
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CAS Number681136-29-8
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分子量365.45
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分子式C19H19N5OS
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纯度98%
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溶解度——
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SMILESO=C(Nc1ccccc1)N1CCN(CC1)c1nc(ns1)c1ccccc1
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化学全称1-Piperazinecarboxamide, N-phenyl-4-(3-phenyl-1,2,4-thiadiazol-5-yl)-
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Karbarz MJ, et al. Anesth Analg, 2009, 108(1), 316-329.
产品手册
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