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Flupirtine
CAS No. 56995-20-1
Flupirtine ( D-9998 )
产品货号. M15076 CAS No. 56995-20-1
A selective neuronal potassium channel (KCNQ/KV7 channel) activator that also has indirect NMDA receptor antagonist and GABAA receptor modulatory properties.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥7857 | 有现货 |
|
| 50MG | ￥16038 | 有现货 |
|
| 100MG | ￥20250 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Flupirtine
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述A selective neuronal potassium channel (KCNQ/KV7 channel) activator that also has indirect NMDA receptor antagonist and GABAA receptor modulatory properties.
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产品描述A selective neuronal potassium channel (KCNQ/KV7 channel) activator that also has indirect NMDA receptor antagonist and GABAA receptor modulatory properties; a centrally acting non-opioid analgesic used as an analgesic for acute and chronic pain.Pain Discontinued
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同义词D-9998
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通路Cell Cycle/DNA Damage
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靶点Potassium Channel
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受体Potassium Channel
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研究领域Neurological Disease
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适应症Pain
化学信息
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CAS Number56995-20-1
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分子量304.32
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分子式C15H17FN4O2
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纯度>98% (HPLC)
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溶解度10 mM in DMSO
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SMILESCCOC(=O)NC1=C(N=C(C=C1)NCC2=CC=C(C=C2)F)N
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化学全称Carbamic acid, N-[2-amino-6-[[(4-fluorophenyl)methyl]amino]-3-pyridinyl]-, ethyl ester
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Szelenyi I, et al. Inflamm Res. 2013 Mar;62(3):251-8.
2. Harish S, et al. J Anaesthesiol Clin Pharmacol. 2012 Apr;28(2):172-7.
3. Hedegaard ER, et al. J Pharmacol Exp Ther. 2016 Apr;357(1):94-102.
2. Harish S, et al. J Anaesthesiol Clin Pharmacol. 2012 Apr;28(2):172-7.
3. Hedegaard ER, et al. J Pharmacol Exp Ther. 2016 Apr;357(1):94-102.
产品手册
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