Potent endogenous ligand of the kisspeptin receptor (KISS1, GPR54). Binds with high affinity to rat and human KISS1 receptors with Ki values of 1.80 and 1.45 nM respectively. Inhibits chemotaxis, invasion and metastasis of human melanomas and breast carcinomas. Stimulates gonadotropin secretion following i.c.v. administration.

天麻素是从中药天麻中提取的一种抗炎多酚，对神经退行性疾病有疗效。

麦考酚酸葡萄糖醛酸是人血浆中麦考酚酸的葡萄糖醛酸代谢产物。