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Entospletinib
CAS No. 1229208-44-9
Entospletinib ( Entospletinib; GS9973; GS 9973 )
产品货号. M17895 CAS No. 1229208-44-9
Entospletinib （IC50= 7.7 nM）is a specific Syk inhibitor, which is orally bioavailable.
纯度: 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥365 | 有现货 |
|
| 5MG | ￥599 | 有现货 |
|
| 10MG | ￥794 | 有现货 |
|
| 25MG | ￥1442 | 有现货 |
|
| 50MG | ￥2203 | 有现货 |
|
| 100MG | ￥3548 | 有现货 |
|
| 200MG | ￥5257 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Entospletinib
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Entospletinib （IC50= 7.7 nM）is a specific Syk inhibitor, which is orally bioavailable.
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产品描述Entospletinib, also known as GS-9973, is a highly selective and orally efficacious Syk inhibitor which is currently undergoing clinical evaluation for autoimmune and oncology indications. In Phase II clinical trials, Entospletinib demonstrates clinical activity in subjects with relapsed or refractory CLL with acceptable toxicity.
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同义词Entospletinib; GS9973; GS 9973
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通路GPCR/G Protein
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靶点Antibacterial
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受体Syk
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研究领域Cancer
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适应症——
化学信息
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CAS Number1229208-44-9
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分子量411.47
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分子式C23H21N7O
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纯度98%
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溶解度DMSO : ≥ 43 mg/mL; 104.51 mM
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SMILESC1CN(CCO1)c1ccc(Nc2nc(cn3ccnc23)c2ccc3cn[nH]c3c2)cc1
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化学全称6-(1H-indazol-6-yl)-N-(4-morpholinophenyl)imidazo[1,2-a]pyrazin-8-amine
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
产品手册
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