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Emodepside

CAS No. 155030-63-0

Emodepside ( PF 1022-221;PF1022-221;BAY 44-4400;BAY44-4400 )

产品货号. M12201 CAS No. 155030-63-0

A semisynthetic derivative of PF1022A, and novel cyclo-depsipeptide anthelmintic which is efficacious against a variety of gastrointestinal nematodes.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
2MG ¥608 有现货
5MG ¥948 有现货
10MG ¥1450 有现货
25MG ¥2665 有现货
50MG ¥4625 有现货
100MG ¥6634 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    Emodepside
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    A semisynthetic derivative of PF1022A, and novel cyclo-depsipeptide anthelmintic which is efficacious against a variety of gastrointestinal nematodes.
  • 产品描述
    A semisynthetic derivative of PF1022A, and novel cyclo-depsipeptide anthelmintic which is efficacious against a variety of gastrointestinal nematodes; causes parasitic nematode muscle relaxation, inhibition of muscle contraction elicited by either ACh or the neuropeptide AF2; elicits a Ca(++)-dependent hyperpolarization of muscle cells.Parasite Infection Phase 1 Clinical
  • 同义词
    PF 1022-221;PF1022-221;BAY 44-4400;BAY44-4400
  • 通路
    Microbiology/Virology
  • 靶点
    Parasite
  • 受体
    Parasite
  • 研究领域
    Infection
  • 适应症
    Parasite Infection

化学信息

  • CAS Number
    155030-63-0
  • 分子量
    1119.39
  • 分子式
    C60H90N6O14
  • 纯度
    >98% (HPLC)
  • 溶解度
    DMSO: ≥ 31 mg/mL
  • SMILES
    O=C([C@H](CC(C)C)N(C)C([C@@H](C)OC([C@H](CC(C)C)N(C)C([C@@H](CC1=CC=C(N2CCOCC2)C=C1)OC([C@H](CC(C)C)N(C)C([C@@H](C)OC([C@H](CC(C)C)N3C)=O)=O)=O)=O)=O)=O)O[C@H](CC4=CC=C(N5CCOCC5)C=C4)C3=O
  • 化学全称
    Cyclo[(αR)-α-hydroxy-4-(4-morpholinyl)benzenepropanoyl-N-methyl-L-leucyl-(2R)-2-hydroxypropanoyl-N-methyl-L-leucyl-(αR)-α-hydroxy-4-(4-morpholinyl)benzenepropanoyl-N-methyl-L-leucyl-(2R)-2-hydroxypropanoyl-N-methyl-L-leucyl]

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1. Harder A, Parasitol Res. 2001 Nov;87(11):924-8.
2. Harder A, et al. Parasitol Res. 2002 Jun;88(6):481-8.
3. Willson J, et al. Parasitology. 2003 Jan;126(Pt 1):79-86.
4. Harder A, et al. Int J Antimicrob Agents. 2003 Sep;22(3):318-31.
产品手册
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