Emodepside
CAS No. 155030-63-0
Emodepside ( PF 1022-221;PF1022-221;BAY 44-4400;BAY44-4400 )
产品货号. M12201 CAS No. 155030-63-0
A semisynthetic derivative of PF1022A, and novel cyclo-depsipeptide anthelmintic which is efficacious against a variety of gastrointestinal nematodes.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥608 | 有现货 |
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5MG | ¥948 | 有现货 |
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10MG | ¥1450 | 有现货 |
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25MG | ¥2665 | 有现货 |
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50MG | ¥4625 | 有现货 |
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100MG | ¥6634 | 有现货 |
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200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称Emodepside
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述A semisynthetic derivative of PF1022A, and novel cyclo-depsipeptide anthelmintic which is efficacious against a variety of gastrointestinal nematodes.
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产品描述A semisynthetic derivative of PF1022A, and novel cyclo-depsipeptide anthelmintic which is efficacious against a variety of gastrointestinal nematodes; causes parasitic nematode muscle relaxation, inhibition of muscle contraction elicited by either ACh or the neuropeptide AF2; elicits a Ca(++)-dependent hyperpolarization of muscle cells.Parasite Infection Phase 1 Clinical
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同义词PF 1022-221;PF1022-221;BAY 44-4400;BAY44-4400
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通路Microbiology/Virology
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靶点Parasite
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受体Parasite
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研究领域Infection
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适应症Parasite Infection
化学信息
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CAS Number155030-63-0
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分子量1119.39
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分子式C60H90N6O14
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纯度>98% (HPLC)
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溶解度DMSO: ≥ 31 mg/mL
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SMILESO=C([C@H](CC(C)C)N(C)C([C@@H](C)OC([C@H](CC(C)C)N(C)C([C@@H](CC1=CC=C(N2CCOCC2)C=C1)OC([C@H](CC(C)C)N(C)C([C@@H](C)OC([C@H](CC(C)C)N3C)=O)=O)=O)=O)=O)=O)O[C@H](CC4=CC=C(N5CCOCC5)C=C4)C3=O
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化学全称Cyclo[(αR)-α-hydroxy-4-(4-morpholinyl)benzenepropanoyl-N-methyl-L-leucyl-(2R)-2-hydroxypropanoyl-N-methyl-L-leucyl-(αR)-α-hydroxy-4-(4-morpholinyl)benzenepropanoyl-N-methyl-L-leucyl-(2R)-2-hydroxypropanoyl-N-methyl-L-leucyl]
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Harder A, Parasitol Res. 2001 Nov;87(11):924-8.
2. Harder A, et al. Parasitol Res. 2002 Jun;88(6):481-8.
3. Willson J, et al. Parasitology. 2003 Jan;126(Pt 1):79-86.
4. Harder A, et al. Int J Antimicrob Agents. 2003 Sep;22(3):318-31.
2. Harder A, et al. Parasitol Res. 2002 Jun;88(6):481-8.
3. Willson J, et al. Parasitology. 2003 Jan;126(Pt 1):79-86.
4. Harder A, et al. Int J Antimicrob Agents. 2003 Sep;22(3):318-31.
产品手册
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