ERAP1-IN-1
CAS No. 865273-97-8
ERAP1-IN-1 ( —— )
产品货号. M26205 CAS No. 865273-97-8
ERAP1-IN-1 is an endoplasmic reticulum aminopeptidase 1 (ERAP1) inhibitor. ERAP1-IN-1 competitively inhibits ERAP1 activity towards a nonamer peptide representative of physiological substrates.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥2341 | 有现货 |
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10MG | ¥3872 | 有现货 |
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25MG | ¥6391 | 有现货 |
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50MG | ¥8748 | 有现货 |
|
100MG | ¥11988 | 有现货 |
|
500MG | ¥24057 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称ERAP1-IN-1
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述ERAP1-IN-1 is an endoplasmic reticulum aminopeptidase 1 (ERAP1) inhibitor. ERAP1-IN-1 competitively inhibits ERAP1 activity towards a nonamer peptide representative of physiological substrates.
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产品描述ERAP1-IN-1 is an endoplasmic reticulum aminopeptidase 1 (ERAP1) inhibitor. ERAP1-IN-1 competitively inhibits ERAP1 activity towards a nonamer peptide representative of physiological substrates.(In Vitro):ERAP1-IN-1 (50 μM) exhibits specific inhibition of ERAP1 in the cellular context. ERAP1-IN-1 allosterically activates ERAP1’s hydrolysis of fluorogenic and chromogenic amino acid substrates.
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同义词——
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通路Others
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靶点Other Targets
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受体Androgen Receptor
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研究领域——
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适应症——
化学信息
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CAS Number865273-97-8
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分子量458.5
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分子式C20H21F3N2O5S
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纯度>98% (HPLC)
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溶解度——
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SMILESCOc1ccc(cc1S(=O)(=O)Nc1cc(ccc1N1CCCCC1)C(F)(F)F)C(O)=O
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Coss CC, Bauler M, Narayanan R, Miller DD, Dalton JT. Alanine aminotransferase regulation by androgens in non-hepatic tissues. Pharm Res. 2012 Apr;29(4):1046-56.
产品手册
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