芦荟素和芦荟大黄素是体外抑制 c-ADH 和 c-ALDH 活性的有效成分。

ACTH (1-17), an adrenocorticotropin analogue, is a potent human melanocortin 1 (MC1) receptor agonist with a Ki of 0.21 nM. Adrenocorticotropic hormone (ACTH), also known as corticotropin, is produced and secreted by the anterior pituitary gland.

NS-2028 是一种高选择性可溶性鸟苷酸环化酶 (sGC) 抑制剂（IC50：基础酶活性和 NO 刺激酶活性分别为 30 nM 和 200 nM）。