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Contezolid
CAS No. 1112968-42-9
Contezolid ( MRX I )
产品货号. M10415 CAS No. 1112968-42-9
Contezolid (MRX I) is an orally active oxazolidinone agent with antibacterial activity Gram-positive pathogens, including MRSA, penicillin-PRSP, PISP, and vancomycin-resistant enterococci (VRE) with MIC of 0.25-4 ug/mL.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥5378 | 有现货 |
|
| 50MG | ￥22518 | 有现货 |
|
| 100MG | ￥29970 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Contezolid
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Contezolid (MRX I) is an orally active oxazolidinone agent with antibacterial activity Gram-positive pathogens, including MRSA, penicillin-PRSP, PISP, and vancomycin-resistant enterococci (VRE) with MIC of 0.25-4 ug/mL.
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产品描述Contezolid (MRX I) is an orally active oxazolidinone agent with antibacterial activity Gram-positive pathogens, including MRSA, penicillin-PRSP, PISP, and vancomycin-resistant enterococci (VRE) with MIC of 0.25-4 ug/mL; demonstrates the same or better efficacy than linezolid in both systemic and local infection models against the tested strains.Bacterial Infection Phase 3 Clinical
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同义词MRX I
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通路GPCR/G Protein
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靶点Antibacterial
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受体Antibacterial
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研究领域Infection
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适应症Bacterial Infection
化学信息
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CAS Number1112968-42-9
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分子量408.34
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分子式C18H15F3N4O4
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纯度>98% (HPLC)
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溶解度——
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SMILESO=C1CCN(C2=C(F)C=C(N3C(O[C@@H](CNC4=NOC=C4)C3)=O)C(F)=C2F)C=C1
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化学全称1-{2,3,6-trifluoro-4-[(5S)-5-{[(1,2-oxazol-3-yl)amino]methyl}-2-oxo-1,3-oxazolidin-3-yl]phenyl}-2,3-dihydropyridin-4(1H)-one
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Li CR, et al. Antimicrob Agents Chemother. 2014;58(4):2418-21.
2. Gordeev MF, et al. J Med Chem. 2014 Jun 12;57(11):4487-97.
3. Meng J, et al. Drug Metab Dispos. 2015 May;43(5):646-59.
4. Eckburg PB, et al. Antimicrob Agents Chemother. 2017 Mar 24;61(4). pii: e02181-16.
2. Gordeev MF, et al. J Med Chem. 2014 Jun 12;57(11):4487-97.
3. Meng J, et al. Drug Metab Dispos. 2015 May;43(5):646-59.
4. Eckburg PB, et al. Antimicrob Agents Chemother. 2017 Mar 24;61(4). pii: e02181-16.
产品手册
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