
Cetrorelix
CAS No. 145672-81-7
Cetrorelix ( —— )
产品货号. M20166 CAS No. 145672-81-7
Cetrorelix Acetate 是促性腺激素释放激素 (GnRH) 受体拮抗剂,IC50 为 1.21 nM。
纯度: >98% (HPLC)






规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥551 | 有现货 |
![]() ![]() |
5MG | ¥778 | 有现货 |
![]() ![]() |
10MG | ¥1312 | 有现货 |
![]() ![]() |
25MG | ¥2738 | 有现货 |
![]() ![]() |
50MG | ¥4512 | 有现货 |
![]() ![]() |
100MG | ¥6415 | 有现货 |
![]() ![]() |
200MG | 获取报价 | 有现货 |
![]() ![]() |
500MG | 获取报价 | 有现货 |
![]() ![]() |
1G | 获取报价 | 有现货 |
![]() ![]() |
生物学信息
-
产品名称Cetrorelix
-
注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
-
产品简述Cetrorelix Acetate 是促性腺激素释放激素 (GnRH) 受体拮抗剂,IC50 为 1.21 nM。
-
产品描述Cetrorelix Acetate is gonadotropin-releasing hormone?(GnRH)?receptor antagonist with an?IC50?of 1.21 nM.(In Vitro):Cetrorelix Acetate inhibits growth of ES-2 cell line at 1000 ng/ml. Cetrorelix Acetate has comparable antiproliferative effects as GnRH-I agonists indicating that the dichotomy of GnRH-I agonists and antagonists might not apply to the GnRH-I system in cancer cells.
-
体外实验Cetrorelix Acetate inhibits growth of ES-2 cell line at 1000 ng/ml. Cetrorelix Acetate has comparable antiproliferative effects as GnRH-I agonists indicating that the dichotomy of GnRH-I agonists and antagonists might not apply to the GnRH-I system in cancer cells.
-
体内实验——
-
同义词——
-
通路Others
-
靶点Other Targets
-
受体GNRHR
-
研究领域Others
-
适应症——
化学信息
-
CAS Number145672-81-7
-
分子量1491.11
-
分子式C70H92ClN17O14.C2H4O2
-
纯度>98% (HPLC)
-
溶解度DMSO:50 mg/mL?(33.53 mM)
-
SMILESCC(O)=O.CC(C)C[C@H](NC(=O)[C@@H](CCCNC(N)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CO)NC(=O)[C@@H](Cc1cccnc1)NC(=O)[C@@H](Cc1ccc(Cl)cc1)NC(=O)[C@@H](Cc1ccc2ccccc2c1)NC(C)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N1CCC[C@H]1C(=O)N[C@H](C)C(N)=O
-
化学全称(S)-1-(((R)-2-((S)-2-((S)-2-((R)-2-((R)-2-((R)-2-acetamido-3-(naphthalen-2-yl)propanamido)-3-(4-chlorophenyl)propanamido)-3-(pyridin-3-yl)propanamido)-3-hydroxypropanamido)-3-(4-hydroxyphenyl)propanamido)-5-ureidopentanoyl)-L-leucyl-L-arginyl)-N-((R)-1-amino-1-oxopropan-2-yl)pyrrolidine-2-carboxamide acetate
运输与储存
-
储存条件(-20℃)
-
运输条件With Ice Pack
-
稳定性≥ 2 years
参考文献
1.Gründker Carsten Emons Günter. Role of gonadotropin-releasing hormone (GnRH) in ovarian cancer[J]. Reproductive Biology & Endocrinology Rb & E 2003 1(1):65-65.
产品手册




关联产品
-
Exendin derivative 1
Exendin derivative 1 is a 39 amino acid peptide.
-
(+)-JQ1 PA
(+)-JQ1 PA 是 Bromodomain 和末端外 (BET) 抑制剂 JQ1 的衍生物,IC50 为 10.4 nM。
-
Dicloxacillin Sodium
双氯西林是一种与苯唑西林相似的耐β-内酰胺酶青霉素,对革兰氏阳性/阴性需氧菌和厌氧菌具有活性。