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CITCO

CAS No. 338404-52-7

CITCO ( —— )

产品货号. M24287 CAS No. 338404-52-7

CITCO inhibits growth and expansion of brain tumour stem cells (BTSCs) and has an EC50 of 49?nM over pregnane X receptor (PXR), and no activity on other nuclear receptors.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥462 有现货
10MG ¥737 有现货
25MG ¥1345 有现货
50MG ¥2155 有现货
100MG ¥3216 有现货
200MG ¥4836 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    CITCO
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    CITCO inhibits growth and expansion of brain tumour stem cells (BTSCs) and has an EC50 of 49?nM over pregnane X receptor (PXR), and no activity on other nuclear receptors.
  • 产品描述
    CITCO inhibits growth and expansion of brain tumour stem cells (BTSCs) and has an EC50 of 49?nM over pregnane X receptor (PXR), and no activity on other nuclear receptors. CITCO is an imidazothiazole derivative and it also is a selective Constitutive androstane receptor (CAR) agonist.
  • 同义词
    ——
  • 通路
    Others
  • 靶点
    Other Targets
  • 受体
    CAR;PXR
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    338404-52-7
  • 分子量
    436.7
  • 分子式
    C19H12Cl3N3OS
  • 纯度
    >98% (HPLC)
  • 溶解度
    DMSO:soluble; H2O:insoluble
  • SMILES
    Clc(cc1)ccc1-c1c(/C=N/OCc(cc2)cc(Cl)c2Cl)n(ccs2)c2n1
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Chakraborty S, et al. Constitutive androstane receptor agonist CITCO inhibits growth and expansion of brain tumour stem cells. Br J Cancer. 2011 Feb 1;104(3):448-59.
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