BIBF0775
CAS No. 334951-90-5
BIBF0775 ( —— )
产品货号. M20053 CAS No. 334951-90-5
BIBF0775 is a selective TGFβ type I receptor (Alk5) inhibitor (IC50: 34 nM).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥1191 | 有现货 |
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10MG | ¥1847 | 有现货 |
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25MG | ¥3062 | 有现货 |
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50MG | ¥4301 | 有现货 |
|
100MG | ¥6221 | 有现货 |
|
500MG | ¥12798 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称BIBF0775
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述BIBF0775 is a selective TGFβ type I receptor (Alk5) inhibitor (IC50: 34 nM).
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产品描述BIBF0775 is a selective TGFβ type I receptor (Alk5) inhibitor (IC50: 34 nM).
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同义词——
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通路Others
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靶点Other Targets
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受体TGFβR1(ALK5);Alk5
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研究领域——
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适应症——
化学信息
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CAS Number334951-90-5
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分子量494.64
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分子式C31H34N4O2
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纯度>98% (HPLC)
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溶解度DMSO: 60 mg/mL
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SMILESCCN(C)C(=O)c1ccc2c(NC(=O)\C2=C(/Nc2ccc(CN3CCCCC3)cc2)c2ccccc2)c1
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化学全称(3Z)-N-Ethyl-23-dihydro-N-methyl-2-oxo-3-[phenyl[[4-(1-piperidinylmethyl)phenyl]amino]methylene]-1H-indole-6-carboxamide
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Roth GJ et al. Design synthesis and evaluation of indolinones as inhibitors of the transforming growth factor β receptor I (TGFβRI). J Med Chem. 2010 Oct 28;53(20):7287-95.
产品手册
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