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BIBF0775

CAS No. 334951-90-5

BIBF0775 ( —— )

产品货号. M20053 CAS No. 334951-90-5

BIBF0775 is a selective TGFβ type I receptor (Alk5) inhibitor (IC50: 34 nM).

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥1191 有现货
10MG ¥1847 有现货
25MG ¥3062 有现货
50MG ¥4301 有现货
100MG ¥6221 有现货
500MG ¥12798 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    BIBF0775
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    BIBF0775 is a selective TGFβ type I receptor (Alk5) inhibitor (IC50: 34 nM).
  • 产品描述
    BIBF0775 is a selective TGFβ type I receptor (Alk5) inhibitor (IC50: 34 nM).
  • 同义词
    ——
  • 通路
    Others
  • 靶点
    Other Targets
  • 受体
    TGFβR1(ALK5);Alk5
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    334951-90-5
  • 分子量
    494.64
  • 分子式
    C31H34N4O2
  • 纯度
    >98% (HPLC)
  • 溶解度
    DMSO: 60 mg/mL
  • SMILES
    CCN(C)C(=O)c1ccc2c(NC(=O)\C2=C(/Nc2ccc(CN3CCCCC3)cc2)c2ccccc2)c1
  • 化学全称
    (3Z)-N-Ethyl-23-dihydro-N-methyl-2-oxo-3-[phenyl[[4-(1-piperidinylmethyl)phenyl]amino]methylene]-1H-indole-6-carboxamide

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Roth GJ et al. Design synthesis and evaluation of indolinones as inhibitors of the transforming growth factor β receptor I (TGFβRI). J Med Chem. 2010 Oct 28;53(20):7287-95.
产品手册
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