AGI-1067 (Succinobucol) 是 TNF-α 诱导的 VCAM-1、MCP-1 和 E-选择素表达的有效抑制剂 (IC50=6,10 和 25 uM)。

Taccalonolide AJ is a microtubule stabilizer; it has excellent and highly persistent antitumor efficacy when administered directly to the tumor, suggesting that the lack of antitumor efficacy seen with systemic administration of AJ is likely due to its short half-life in vivo.

Ilmetropium iodide 是一种支气管扩张剂。