Atipamezole
CAS No. 104054-27-5
Atipamezole ( MPV-1248;MPV1248;MPV 1248 )
产品货号. M10207 CAS No. 104054-27-5
Antipamezole (MPV-1248) is a potent, specific α2-adrenoceptor antagonist with Ki of 1.6 nM.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥389 | 有现货 |
|
10MG | ¥551 | 有现货 |
|
25MG | ¥1158 | 有现货 |
|
50MG | ¥2041 | 有现货 |
|
100MG | ¥3062 | 有现货 |
|
200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
-
产品名称Atipamezole
-
注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
-
产品简述Antipamezole (MPV-1248) is a potent, specific α2-adrenoceptor antagonist with Ki of 1.6 nM.
-
产品描述Antipamezole (MPV-1248) is a potent, specific α2-adrenoceptor antagonist with Ki of 1.6 nM; reverses the effects of the sedative dexmedetomidine and medetomidine as a veterinary drug.Alcoholism Phase 1 Discontinued
-
同义词MPV-1248;MPV1248;MPV 1248
-
通路Angiogenesis
-
靶点Adrenergic Receptor
-
受体α2-adrenoceptor
-
研究领域Neurological Disease
-
适应症Alcoholism
化学信息
-
CAS Number104054-27-5
-
分子量212.29
-
分子式C14H16N2
-
纯度>98% (HPLC)
-
溶解度DMSO: ≥30 mg/mL
-
SMILESCCC1(C2=CNC=N2)CC3=C(C=CC=C3)C1
-
化学全称1H-Imidazole, 5-(2-ethyl-2,3-dihydro-1H-inden-2-yl)-
运输与储存
-
储存条件(-20℃)
-
运输条件With Ice Pack
-
稳定性≥ 2 years
参考文献
1. Pertovaara A, et al. CNS Drug Rev. 2005 Autumn;11(3):273-88.
2. Scheinin H, et al. Eur J Pharmacol. 1988 Jun 22;151(1):35-42.
3. Scheinin H, et al. Eur J Pharmacol. 1986 Sep 23;129(1-2):113-21.
4. Karhuvaara S, et al. Br J Clin Pharmacol. 1990 Jul;30(1):97-106.
2. Scheinin H, et al. Eur J Pharmacol. 1988 Jun 22;151(1):35-42.
3. Scheinin H, et al. Eur J Pharmacol. 1986 Sep 23;129(1-2):113-21.
4. Karhuvaara S, et al. Br J Clin Pharmacol. 1990 Jul;30(1):97-106.
产品手册
关联产品
-
Dicentrine
Dicentrine is a natural product isolated from the plant Lindera megaphylla with antihypertensive effect. Dicentrine is an α1-adrenoceptor antagonist which has effective against human hyperplastic prostates.
-
BRL 44408 maleate
A potent, selective α2A-adrenoceptor antagonist with Ki of 1.7 nM, 80-fold selectivity over α2B-adrenergic receptors.
-
Guanfacine hydrochlo...
A selective α2A receptor agonist that can reduce peripheral sympathetic outflow and thus cansues a reduction in peripheral sympathetic tone.