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Atipamezole

CAS No. 104054-27-5

Atipamezole ( MPV-1248;MPV1248;MPV 1248 )

产品货号. M10207 CAS No. 104054-27-5

Antipamezole (MPV-1248) is a potent, specific α2-adrenoceptor antagonist with Ki of 1.6 nM.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥389 有现货
10MG ¥551 有现货
25MG ¥1158 有现货
50MG ¥2041 有现货
100MG ¥3062 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    Atipamezole
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Antipamezole (MPV-1248) is a potent, specific α2-adrenoceptor antagonist with Ki of 1.6 nM.
  • 产品描述
    Antipamezole (MPV-1248) is a potent, specific α2-adrenoceptor antagonist with Ki of 1.6 nM; reverses the effects of the sedative dexmedetomidine and medetomidine as a veterinary drug.Alcoholism Phase 1 Discontinued
  • 同义词
    MPV-1248;MPV1248;MPV 1248
  • 通路
    Angiogenesis
  • 靶点
    Adrenergic Receptor
  • 受体
    α2-adrenoceptor
  • 研究领域
    Neurological Disease
  • 适应症
    Alcoholism

化学信息

  • CAS Number
    104054-27-5
  • 分子量
    212.29
  • 分子式
    C14H16N2
  • 纯度
    >98% (HPLC)
  • 溶解度
    DMSO: ≥30 mg/mL
  • SMILES
    CCC1(C2=CNC=N2)CC3=C(C=CC=C3)C1
  • 化学全称
    1H-Imidazole, 5-(2-ethyl-2,3-dihydro-1H-inden-2-yl)-

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1. Pertovaara A, et al. CNS Drug Rev. 2005 Autumn;11(3):273-88.
2. Scheinin H, et al. Eur J Pharmacol. 1988 Jun 22;151(1):35-42.
3. Scheinin H, et al. Eur J Pharmacol. 1986 Sep 23;129(1-2):113-21.
4. Karhuvaara S, et al. Br J Clin Pharmacol. 1990 Jul;30(1):97-106.
产品手册
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