Atipamezole
CAS No. 104054-27-5
Atipamezole ( MPV-1248;MPV1248;MPV 1248 )
产品货号. M10207 CAS No. 104054-27-5
Antipamezole (MPV-1248) is a potent, specific α2-adrenoceptor antagonist with Ki of 1.6 nM.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥389 | 有现货 |
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10MG | ¥551 | 有现货 |
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25MG | ¥1158 | 有现货 |
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50MG | ¥2041 | 有现货 |
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100MG | ¥3062 | 有现货 |
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200MG | 获取报价 | 有现货 |
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500MG | 获取报价 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称Atipamezole
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Antipamezole (MPV-1248) is a potent, specific α2-adrenoceptor antagonist with Ki of 1.6 nM.
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产品描述Antipamezole (MPV-1248) is a potent, specific α2-adrenoceptor antagonist with Ki of 1.6 nM; reverses the effects of the sedative dexmedetomidine and medetomidine as a veterinary drug.Alcoholism Phase 1 Discontinued
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同义词MPV-1248;MPV1248;MPV 1248
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通路Angiogenesis
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靶点Adrenergic Receptor
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受体α2-adrenoceptor
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研究领域Neurological Disease
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适应症Alcoholism
化学信息
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CAS Number104054-27-5
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分子量212.29
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分子式C14H16N2
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纯度>98% (HPLC)
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溶解度DMSO: ≥30 mg/mL
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SMILESCCC1(C2=CNC=N2)CC3=C(C=CC=C3)C1
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化学全称1H-Imidazole, 5-(2-ethyl-2,3-dihydro-1H-inden-2-yl)-
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Pertovaara A, et al. CNS Drug Rev. 2005 Autumn;11(3):273-88.
2. Scheinin H, et al. Eur J Pharmacol. 1988 Jun 22;151(1):35-42.
3. Scheinin H, et al. Eur J Pharmacol. 1986 Sep 23;129(1-2):113-21.
4. Karhuvaara S, et al. Br J Clin Pharmacol. 1990 Jul;30(1):97-106.
2. Scheinin H, et al. Eur J Pharmacol. 1988 Jun 22;151(1):35-42.
3. Scheinin H, et al. Eur J Pharmacol. 1986 Sep 23;129(1-2):113-21.
4. Karhuvaara S, et al. Br J Clin Pharmacol. 1990 Jul;30(1):97-106.
产品手册
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