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Artefenomel
CAS No. 1029939-86-3
Artefenomel ( OZ439 )
产品货号. M10144 CAS No. 1029939-86-3
Artefenomel (OZ439) is a novel, next-generation antimalarial ozonide that demonstrates high potentcy against P. falciparum in vitro and P. berghei in vivo (K1/NF54, IC50=2.0/3.2 nM).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥3613 | 有现货 |
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| 50MG | ￥15066 | 有现货 |
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| 100MG | ￥22518 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Artefenomel
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Artefenomel (OZ439) is a novel, next-generation antimalarial ozonide that demonstrates high potentcy against P. falciparum in vitro and P. berghei in vivo (K1/NF54, IC50=2.0/3.2 nM).
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产品描述Artefenomel (OZ439) is a novel, next-generation antimalarial ozonide that demonstrates high potentcy against P. falciparum in vitro and P. berghei in vivo (K1/NF54, IC50=2.0/3.2 nM).Parasite Infection Phase 2 Clinical
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同义词OZ439
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通路Microbiology/Virology
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靶点Parasite
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受体Parasite
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研究领域Infection
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适应症Parasite Infection
化学信息
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CAS Number1029939-86-3
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分子量469.62
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分子式C28H39NO5
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纯度>98% (HPLC)
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溶解度——
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SMILESC1CC2(CCC1C3=CC=C(C=C3)OCCN4CCOCC4)OC5(C6CC7CC(C6)CC5C7)OO2
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化学全称4-[2-(4-cis-Dispiro[cyclohexane-1,3'-[1,2,4]trioxolane-5',2''-tricyclo[3.3.1.13,7]decan]-4-ylphenoxy)ethyl]morpholine
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Dong Y, et al. J Med Chem. 2017 Apr 13;60(7):2654-2668.
2. Kim HS, et al. J Med Chem. 2017 Apr 13;60(7):2651-2653.
3. Macintyre F, et al. BMC Med. 2017 Oct 9;15(1):181.
4. Yang T, et al. Antimicrob Agents Chemother. 2016 Jul 22;60(8):4501-10.
2. Kim HS, et al. J Med Chem. 2017 Apr 13;60(7):2651-2653.
3. Macintyre F, et al. BMC Med. 2017 Oct 9;15(1):181.
4. Yang T, et al. Antimicrob Agents Chemother. 2016 Jul 22;60(8):4501-10.
产品手册
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